DMPX
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| Identifiers | |
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| CAS Number | 14114-46-6  |
| ATC code | None |
| PubChem | CID 99562 |
| Chemical data | |
| Formula | C10H10N4O2 |
| Molar mass | 218.212 g/mol |
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DMPX (3,7-Dimethyl-1-propargylxanthine) is a caffeine analog which displays affinity to A2-adenosine receptors, in contrast to the A1 subtype receptors.[1] DMPX had 28× & 15× higher potency than caffeine in blocking peripheral and central NECA-responses. The locomotor stimulation caused by DMPX (ED50 10 μmol/kg) was similarly higher than caffeine.[1]
References[edit]
- ^ a b 3,7-Dimethyl-1-propargylxanthine: a potent and selective in vivo antagonist of adenosine analogs. Life Sci. 1988;43(21):1671-84. PMID 3193854
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